Setidegrasib
Pharmaceutical compound

Setidegrasib is an investigational new drug that is being evaluated by Astellas Pharma for the treatment of solid tumors. It is an PROTACs degrader of the KRAS protein harboring a G12D mutation.
01Clinical trials
Setidegrasib in combination with either FOLFIRINOX or NALIRIFOX chemotherapy is currently in phase 3 clinical trials for the treatment of pancreatic cancer.
Sources and credits
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- Setidegrasib.svg by Boghog, CC0
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